GPCR化合物庫- Medchemexpress (MCE)

1、標(biāo)題：GPCR化合物庫- Medchemexpress （MCE）品牌： Medchemexpress （MCE）保存條件： -20供應(yīng)商： MCE中國數(shù)量： 大量保質(zhì)期： 2年規(guī)格：提供組合定制服務(wù)（現(xiàn)貨供應(yīng)）供貨地址：美國     MedChemExpress (MCE)專注于各種抑制劑、調(diào)節(jié)劑、API、天然產(chǎn)物及化合物庫，總部位于美國新澤西。MCE經(jīng)過十年努力已成為全球生物活性小分子領(lǐng)域的一流供應(yīng)商。MedChemExpress(MCE)產(chǎn)品涵蓋近20個熱門研究領(lǐng)域，1000多個細分靶點，超過3000個現(xiàn)貨抑制劑、拮抗劑和激動劑。相關(guān)的應(yīng)用成果已發(fā)表于Nat

2、ure、Cell等國際知名雜志，在全球20余個國家地區(qū)設(shè)有代理機構(gòu)。上海皓元生物醫(yī)藥科技有限公司(MCE 中國) 是MedChemExpress (MCE) 亞洲總代理。  貨號：HY-L006 A unique collection of 190 small molecules targeting G protein coupled receptors used in GPCR screening for various research and drug development projects. All of the small molecules in the GPCR li

3、brary are well characterized with biological and pharmaceutical activity. A powerful tool for discovering GPCR-based drugs that are the richest signal receptor targets for drug discovery. Targets such as 5-HT Receptor, Dopamine Receptor, Opioid Receptor, Adrenergic Receptors, Cannabinoid Receptor, m

4、GluR, and ETA-receptor etc. Structurally diverse, medicinally active, and cell permeable. Rich documentation with structure, IC50, and brief introduction. NMR and HPLC validated to ensure the highest purity.Formulation: A collection of 190 active molecules supplied as pre-dissolved DMSO solutio

5、nsContainer: 96 Well Format Sample Storage Tube With Screw Cap and Optional 2D BarcodeStability: 3 months -20°C in DMSO, 6 months -80°C in DMSOShipping: Blue icePackaging: Inert gasPlate layout: HY-EmptyAlosetron (Hydrochloride)AripiprazoleBRL 54443Clozapin

6、e N-oxideCP-809101 (hydrochloride)bEmptyOndansetron (hydrochloride dihydrate)Palonosetron (Hydrochloride)QuetiapineSB 271046 (Hydrochloride)SB-269970 (hydrochloride)cEmptyWAY-100635 (maleate salt)AdoprazineCapadenosonIstradefyllineLUF6000dEmptyHOKU-81ICI 118,551 (hydrochloride)IndacaterolIsoprenalin

7、e (hydrochloride)Ivabradine (hydrochloride)eEmptyTapentadol (hydrochloride)Angiotensin II humanAVE 0991AzilsartanAzilsartan medoxomil (monopotassium)fEmptyAM630JWH 073OtenabantRimonabant (Hydrochloride)TaranabantgEmptyINCB3344MK-0812MK-0974MK-3207 (Hydrochloride)OlcegepanthEmptySCH 527123SCH 546738S

8、CH 563705SRT3190WZ811789101112aLorcaserin (Hydrochloride)LoxapineLu AE58054 (Hydrochloride)LY 344864OlanzapineEmptybSB-742457SetiptilineTianeptineTropisetronVortioxetineEmptycPreladenantTozadenantAdipoRonCarvedilolFormoterol (Fumarate)EmptydMirabegronSalmeterol xinafoateSilodosinVilanterolAsenapineE

9、mptyeEprosartan (mesylate)OlmesartanOlmesartan medoxomilPD 123319 (ditrifluoroacetate)TelmisartanEmptyfWIN 55,212-2 (Mesylate)Calcium-Sensing Receptor Antagonists ICinacalcetNPS-2143NPS-2143 (hydrochloride)EmptygAMD-070 (hydrochloride)AMG 487NBI-74330PlerixaforReparixinEmptyhAMD 3465 (hexahydrobromi

10、de)Lurasidone (Hydrochloride)AmisulprideArmodafinilBrexpiprazoleEmptyPlate layout: HY-EmptyCariprazineHaloperidolPaliperidonerac-Rotigotine (Hydrochloride)RotigotinebEmptyBosentanMacitentanSitaxsentan (sodium)ZibotentanAnamorelincEmptyMK 0893BudesonideCortisone (acetate)DexamethasoneGlu

11、cocorticoid receptor agonistdEmptyGPR120 modulator 2GPR40 Activator 1GW-1100GW9508TAK-875eEmptyEbrotidineLoratadineMetiamidePitolisant (hydrochloride)ZaltidinefEmptyKi16425(R)-(+)-Tolterodine(R)-5-Hydroxymethyl TolterodineAclidinium (Bromide)CevimelinegEmptyUmeclidinium (bromide)VU0152100Xanomeline

12、(oxalate)CTEPDipragluranthEmptyVU 0357121GSK962040AprepitantNKP608SB-222200789101112aST-836 (hydrochloride)Ziprasidone (hydrochloride monohydrate)AmbrisentanAtrasentan (hydrochloride)AvosentanEmptybIbutamoren (Mesylate)Exendin-4glucagon receptor antagonists-1glucagon receptor antagonists-2glucagon r

13、eceptor antagonists-3EmptycTGR5 Receptor AgonistMK-6892GSK1292263MBX-2982GPR120 modulator 1EmptydTUG-770Bavisant (dihydrochloride hydrate)Bepotastine (Beslilate)Ciproxifan (maleate)Clemizole (hydrochloride)EmptyeFenspiride (Hydrochloride)Montelukast (sodium)AM095AM966Fingolimod (hydrochloride)Emptyf

14、DarifenacinDiphenmanil (methylsulfate)Solifenacin (hydrochloride)Tarafenacin (D-tartrate)Tiotropium (Bromide)EmptygLY341495LY404039mGlu2 agonistMPEP (Hydrochloride)MTEP (hydrochloride)EmptyhTalnetantML314ADL-5859Alvimopan (dihydrate)BAN ORL 24EmptyPlate layout: HY-EmptyCebranopadolJDTic

15、 (dihydrochloride)Meptazinol (hydrochloride)Methylnaltrexone (Bromide)Naloxone (hydrochloride)bEmptySuvorexantTCS 1102MRS 2578PrasugrelTicagrelorcEmptyProstaglandin E1SalirasibCCG-63802CCG-63808Siramesine (hydrochloride)dEmptyEmptyEmptyEmptyEmptyEmptyeEmptyEmptyEmptyEmptyEmptyEmptyfEmptyEmptyEmptyEmptyEmptyEmptygEmptyEmptyEmptyEmptyEmptyEmptyhEmptyEmptyEmptyEmptyEmptyEmpty789101112aNaltrexoneAlmorexant (hydrochloride)SB-334867 (free base)SB-408124SB-674042EmptybAH 6809LaropiprantMK-2894OC000459ONO-AE3-208Empty